Acetaminophen (paracetamol) + Chlorpheniramine

Indications

Acetaminophen (paracetamol) + Chlorpheniramine is used for: Relief of Cold & Flu Symptoms

Adult Dose

Relief of Cold & Flu Symptoms 2 tablets PO q4hr

Child Dose

Relief of Cold & Flu Symptoms >12 years: 2 tablets PO q4hr

Renal Dose

Administration

Contra Indications

Contraindicated in documented hypersensitivity; asthma attacks, narrow-angle glaucoma, symptomatic prostate hypertrophy, bladder-neck obstruction, and stenosing peptic ulcer; known G-6-PD deficiency Chlorpheniramine may cause significant confusional symptoms; not for administration to premature or full-term neonates Acetaminophen hepatotoxicity possible in chronic alcoholics following various dose levels; severe or recurrent pain or high or continued fever may indicate a serious illness; contained in many OTC products and combined use with these products may result in toxicity due to cumulative doses exceeding recommended maximum dose Acetaminophen: Risk for rare, but serious skin reactions that can be fatal; these reactions include Stevens-Johnson Syndrome (SJS), toxic epidermal necrolysis (TEN), and acute generalized exanthematous pustulosis (AGEP); symptoms may include skin redness, blisters and rash

Precautions

Pregnancy-Lactation

Interactions

Adverse Effects

Side effects of Acetaminophen (paracetamol) + Chlorpheniramine : Hypotension Palpitations Tachycardia Anxiety Confusion Depression Dizziness Drowsiness Euphoria Fatigue Headache Insomnia Irritability Nervousness Tremors Anorexia Constipation Diarrhea Nausea Vomiting Agranulocytosis Anemia Blood dyscrasias (neutropenia, pancytopenia, leukopenia, thrombocytopenia) Hemolytic anemia Bilirubin and alkaline phosphatase may increase Thickening of bronchial secretions Wheezing Dry mouth, nose, throat

Mechanism of Action

Chlorpheniramine blocks muscle responses in histamine and acts as an antagonism of the constrictor effects of histamine on respiratory smooth muscle. Acetaminophen blocks pain impulse generation peripherally and may inhibit the generation of prostaglandin in the CNS. Reduces fever by inhibiting the hypothalamic heat-regulating center.