Lafutidine
Indications
Lafutidine is used for:
Gastric and duodenal ulcers; Stomal ulcers, Gastric mucosal lesions
Adult Dose
Oral
Gastric and duodenal ulcers; Stomal ulcers
Adult: 10 mg bid, once after breakfast, once after evening meal or before sleeping. Adjust dose according to patient's age and symptoms.
Gastric mucosal lesions
Adult: 10 mg once daily, after evening meal or before sleeping. Adjust dose according to patient's age and symptoms.
Pre-anaesthetic medication
Adult: 10 mg before sleeping on the day before operation, and 10 mg 2 hr before introduction of anaesthetic on the day of operation.
Elderly: Dose reduction or increase in dosing interval may be needed.
Hepatic impairment: Dose reduction or increase in dosing interval may be needed.
Child Dose
Renal Dose
Renal impairment: Dose reduction or increase in dosing interval may be needed.
Administration
Contra Indications
Lactation.
Precautions
Hepatic and renal impairment. Elderly.
Pregnancy-Lactation
Interactions
Adverse Effects
Side effects of Lafutidine :
Constipation, hyperuricaemia, increase in LFT and total bilirubin, gynaecomastia, anorexia, hallucinations.
Potentially Fatal: Anaphylactic reactions, blood dyscrasias (e.g. agranulocytosis, thrombocytopenia).
Mechanism of Action
Lafutidine is a histamine H2-antagonist with gastroprotective activity. It is used in the treatment of gastric ulcers and before general anaesthesia to reduce the incidence of aspiration pneumonia.